Khateeta M. Emerson

Process Development of C–N Cross-Coupling and Enantioselective Biocatalytic Reactions for the Asymmetric Synthesis of Niraparib

Cheol K. Chung, Paul G. Bulger, Birgit Kosjek et al. · Organic Process Research & Development · 2013 · 169 citations

Natural Sciences, Chemistry, Medicinal Chemistry +17

Synthesis of a Muscarinic Receptor Antagonist via a Diastereoselective Michael Reaction, Selective Deoxyfluorination and Aromatic Metal−Halogen Exchange Reaction

Toshiaki Mase, Ioannis N. Houpis, Atsushi Akao et al. · The Journal of Organic Chemistry · 2001 · 92 citations

Pharmacy, Chemistry, Medicinal Chemistry +13

Practical Asymmetric Synthesis of Aprepitant, a Potent Human NK-1 Receptor Antagonist, via a Stereoselective Lewis Acid-Catalyzed Trans Acetalization Reaction

Matthew M. Zhao, James M. McNamara, Guo-Jie Ho et al. · The Journal of Organic Chemistry · 2002 · 65 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12

Development of a Fit-for-Purpose Large-Scale Synthesis of an Oral PARP Inhibitor

Debra J. Wallace, Carl A. Baxter, Karel J. M. Brands et al. · Organic Process Research & Development · 2011 · 56 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13

Carbodiimide-Mediated Amide Formation in a Two-Phase System. A High-Yield and Low-Racemization Procedure for Peptide Synthesis

Guo‐Jie Ho, Khateeta M. Emerson, David J. Mathre et al. · The Journal of Organic Chemistry · 1995 · 54 citations

Life Sciences, Biochemistry, Biocatalysis +7