Concepedia

Arnault Massink

AM

Statistics

Publications

8

Citations

398

H-Index

8

Active since

2013

Affiliations

Centre for Human Drug Research(Current)

Leiden University

University of Ferrara

Uppsala University

Scripps Research Institute

Arnault Massink is an author at Centre for Human Drug Research specializing in ligand binding, pharmacology, and molecular pharmacology.

Publications per year

2013–2016

8

Publications

8

The Role of a Sodium Ion Binding Site in the Allosteric Modulation of the A2A Adenosine G Protein-Coupled Receptor

Hugo Gutiérrez‐de‐Terán, Arnault Massink, David Rodríguez et al. · Structure · 2013 · 141 citations · Full text

, , +16

Sodium Ion Binding Pocket Mutations and Adenosine A2A Receptor Function

Arnault Massink, Hugo Gutiérrez‐de‐Terán, Eelke B. Lenselink et al. · Molecular Pharmacology · 2014 · 100 citations · Full text

, , +17

Synthesis and Biological Evaluation of Novel Allosteric Enhancers of the A<sub>1</sub>Adenosine Receptor Based on 2-Amino-3-(4′-Chlorobenzoyl)-4-Substituted-5-Arylethynyl Thiophene

Romeo Romagnoli, Pier Giovanni Baraldi, Adriaan P. IJzerman et al. · Journal of Medicinal Chemistry · 2014 · 32 citations · Full text

, , +17

5′-Substituted Amiloride Derivatives as Allosteric Modulators Binding in the Sodium Ion Pocket of the Adenosine A<sub>2A</sub>Receptor

Arnault Massink, Julien Louvel, Ilze Adlere et al. · Journal of Medicinal Chemistry · 2016 · 31 citations · Full text

, , +17

Molecular mechanism of allosteric modulation at<scp>GPCRs</scp>: insight from a binding kinetics study at the human<scp>A</scp><sub>1</sub>adenosine receptor

Dong Guo, Suzanne N Venhorst, Arnault Massink et al. · British Journal of Pharmacology · 2014 · 28 citations · Full text

, , +17

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