Małgorzata Pawełczak

Structure-Guided, Single-Point Modifications in the Phosphinic Dipeptide Structure Yield Highly Potent and Selective Inhibitors of Neutral Aminopeptidases

Stamatia Vassiliou, Ewelina Węglarz‐Tomczak, Łukasz Berlicki et al. · Journal of Medicinal Chemistry · 2014 · 55 citations · Full text

Bioorganic Chemistry, Alanyl Aminopeptidase, Selective Inhibitors +18

α-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine- and neutral aminopeptidases

Marcin Drąg, Jolanta Grembecka, Małgorzata Pawełczak et al. · European Journal of Medicinal Chemistry · 2005 · 44 citations

Experimental Optimisation, Molecular Pharmacology, Medicinal Chemistry +11

Unnatural amino acids increase activity and specificity of synthetic substrates for human and malarial cathepsin C

Marcin Poręba, Marko Mihelič, Priscilla Krai et al. · Amino Acids · 2013 · 41 citations · Full text

Individual stereoisomers of phosphinic dipeptide inhibitor of leucine aminopeptidase

Artur Mucha, Michael Lämmerhofer, Wolfgang Lindner et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 29 citations · Full text

Medicinal Chemistry, Biochemistry, Natural Sciences +4

A structural insight into the P1 S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases

Ewelina Węglarz‐Tomczak, Łukasz Berlicki, Małgorzata Pawełczak et al. · European Journal of Medicinal Chemistry · 2016 · 28 citations · Full text

Medicinal Chemistry, Biochemistry, P1 S1 +10