Fabrizio Pertusati

Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer

Marcella Bassetto, Salvatore Ferla, Fabrizio Pertusati et al. · European Journal of Medicinal Chemistry · 2016 · 71 citations · Full text

Diastereoselective synthesis of P-chirogenic phosphoramidate prodrugs of nucleoside analogues (ProTides) via copper catalysed reaction

Fabrizio Pertusati, Christopher McGuigan · Chemical Communications · 2015 · 47 citations · Full text

P-chirogenic Phosphoramidate Prodrugs, Engineering, Organic Chemistry +16

ProTides of N-(3-(5-(2′-deoxyuridine))prop-2-ynyl)octanamide as potential anti-tubercular and anti-viral agents

Christopher McGuigan, Marco Derudas, Blanka Gönczy et al. · Bioorganic & Medicinal Chemistry · 2014 · 36 citations · Full text

Medicinal Chemistry, Medicine, Antiviral Drug Development +6

Design, synthesis and biological evaluation of phosphorodiamidate prodrugs of antiviral and anticancer nucleosides

Christopher McGuigan, Claire Bourdin, Marco Derudas et al. · European Journal of Medicinal Chemistry · 2013 · 32 citations · Full text

Medicinal Chemistry, Biochemistry, Medicine +10

Synthesis of an Apionucleoside Family and Discovery of a Prodrug with Anti-HIV Activity

Kiran S. Toti, Marco Derudas, Fabrizio Pertusati et al. · The Journal of Organic Chemistry · 2014 · 31 citations

Anti-hiv Activity, Bioorganic Chemistry, Molecular Biology +20