Vaishali Humnabadkar

Azaindoles: Noncovalent DprE1 Inhibitors from Scaffold Morphing Efforts, Kill Mycobacterium tuberculosis and Are Efficacious <i>in Vivo</i>

Pravin S. Shirude, Radha Krishan Shandil, C Sadler et al. · Journal of Medicinal Chemistry · 2013 · 161 citations

Pharmacotherapy, Antimicrobial Chemotherapy, Pharmaceutical Chemistry +22

4-Aminoquinolone Piperidine Amides: Noncovalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial Activity

Maruti Naik, Vaishali Humnabadkar, Subramanyam J. Tantry et al. · Journal of Medicinal Chemistry · 2014 · 93 citations · Full text

Discovery of Pyrazolopyridones as a Novel Class of Noncovalent DprE1 Inhibitor with Potent Anti-Mycobacterial Activity

Manoranjan Panda, Sreekanth A. Ramachandran, Vasanthi Ramachandran et al. · Journal of Medicinal Chemistry · 2014 · 93 citations

Antimicrobial Chemotherapy, Pharmaceutical Chemistry, Potent Anti-mycobacterial Activity +20

Lead Optimization of 1,4-Azaindoles as Antimycobacterial Agents

Pravin S. Shirude, Radha Krishan Shandil, M. R. Manjunatha et al. · Journal of Medicinal Chemistry · 2014 · 88 citations · Full text

Aminopyrazinamides: Novel and Specific GyrB Inhibitors that Kill Replicating and Nonreplicating <i>Mycobacterium tuberculosis</i>

Pravin S. Shirude, Prashanti Madhavapeddi, Julie A. Tucker et al. · ACS Chemical Biology · 2012 · 86 citations

Crystal Structure, Tuberculosis Prevention, Pharmacotherapy +21