Martin Lochner

Identification of potent and selective small molecule inhibitors of the cation channel <scp>TRPM4</scp>

Lijo Cherian Ozhathil, Clémence Delalande, Beatrice Bianchi et al. · British Journal of Pharmacology · 2018 · 77 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

The muscarinic antagonists scopolamine and atropine are competitive antagonists at 5-HT 3 receptors

Martin Lochner, Andrew J. Thompson · Neuropharmacology · 2016 · 76 citations · Full text

Medicine, Neuroscience, Pharmacology +17

Design, synthesis and pharmacological characterization of analogs of 2-aminoethyl diphenylborinate (2-APB), a known store-operated calcium channel blocker, for inhibition of TRPV6-mediated calcium transport

Alexandre Hofer, Gergely Kovács, Anna Zappatini et al. · Bioorganic & Medicinal Chemistry · 2013 · 61 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16

Selective activation of Gαob by an adenosine A1 receptor agonist elicits analgesia without cardiorespiratory depression

Mark J. Wall, Emily Hill, Robert Huckstepp et al. · Nature Communications · 2022 · 57 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Agonists and Antagonists Bind to an A-A Interface in the Heteromeric 5-HT3AB Receptor

Martin Lochner, Sarah C. R. Lummis · Biophysical Journal · 2010 · 55 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16