Huda Zahid

Selective N‐Terminal BET Bromodomain Inhibitors by Targeting Non‐Conserved Residues and Structured Water Displacement**

Huarui Cui, Anand Divakaran, Anil K. Pandey et al. · Angewandte Chemie International Edition · 2020 · 43 citations · Full text

Molecular Biology, Chemical Biology, Non‐conserved Residues +16

4-Methyl-1,2,3-Triazoles as <i>N</i>-Acetyl-Lysine Mimics Afford Potent BET Bromodomain Inhibitors with Improved Selectivity

Huarui Cui, Angela S. Carlson, Mary A. Schleiff et al. · Journal of Medicinal Chemistry · 2021 · 33 citations · Full text

A Structure-based Design Approach for Generating High Affinity BRD4 D1-Selective Chemical Probes

Huarui Cui, Anand Divakaran, Zachariah J. Hoell et al. · Journal of Medicinal Chemistry · 2022 · 33 citations · Full text

Selectivity, ligand deconstruction, and cellular activity analysis of a BPTF bromodomain inhibitor

Steven E. Kirberger, Peter D. Ycas, Jorden A. Johnson et al. · Organic & Biomolecular Chemistry · 2019 · 31 citations

New Design Rules for Developing Potent Cell-Active Inhibitors of the Nucleosome Remodeling Factor (NURF) via BPTF Bromodomain Inhibition

Huda Zahid, Caroline R. Buchholz, Manjulata Singh et al. · Journal of Medicinal Chemistry · 2021 · 27 citations · Full text