Agonistic and antagonistic properties of the bradykinin B₂ receptor antagonist, Hoe 140, in isolated blood vessels from different species

Michel Félétou, Martine Germain, Christophe Thurieau, +2

British Journal of Pharmacology

Vascular DiseaseCardiovascular PharmacologyPharmacotherapyDifferent SpeciesBradykinin B2 Antagonist +16

A Novel Synthetic Inhibitor of CDC25 Phosphatases

Marie-Christine Brézak, Muriel Quaranta, Odile Mondésert, +11

Cancer Research

Identification of Potent Non-Peptide Somatostatin Antagonists with sst₃ Selectivity

Lydie Poitout, Pierre Roubert, Marie-Odile Contour-Galcéra, +6

Journal of Medicinal Chemistry

Molecular PharmacologyMedicinal ChemistryNon-peptide Somatostatin AnaloguesBiochemistryFunctional Selectivity +13

Link protein interactions with hyaluronate and proteoglycans. Characterization of two distinct domains in bovine cartilage link proteins.

J.-P. Périn, Fabrice Bonnet, Christophe Thurieau, +1

Journal of Biological Chemistry

Protein AssemblyGlycobiologyMolecular BiologyCarbohydrate-protein InteractionMusculoskeletal Research +21

Molecular Cloning and Complete Amino Acid Sequence of AP50, an Assembly Protein Associated with Clathrin-Coated Vesicles

Christophe Thurieau, Jürgen Brosius, CINDY BURNE, +6

DNA

Proteinlipid InteractionAp50 Cdna ClonesProtein FunctionBiochemistryProtein Assembly +12

Novel pharmacological MC4R agonists can efficiently activate mutated MC4R from obese patient with impaired endogenous agonist response

Pierre Roubert, Béatrice Dubern, Pascale Plas, +8

Journal of Endocrinology

Human GrowthMetabolic RemodelingObesityMetabolic SyndromeMolecular Pharmacology +19

The 50 kDa protein subunit of assembly polypeptide (AP) AP-2 adaptor from clathrin-coated vesicles is phosphorylated on threonine-156 by AP-1 and a soluble AP50 kinase which co-purifies with the assembly polypeptides

Alain Pauloin, Christophe Thurieau

Biochemical Journal

Proteinlipid InteractionMolecular BiologySoluble Ap50 KinaseRadioactive PeptideMolecular Pharmacology +15

In vitro effects of HOE 140 in human bronchial and vascular tissue

Michel Félétou, Corinne Martin‐Chouly, Mathiéu Molimard, +6

European Journal of Pharmacology

AsthmaPulmonary CirculationRespiratory ToxicologyMedicineHoe 140 +8

Venous and arterial endothelial cells respond differently to thrombin and its endogenous receptor agonist

Serge Simonet, Edith Bonhomme, Michel Laubie, +3

European Journal of Pharmacology

ThrombosisVenous DiseaseSignal TransductionVenous ThrombosisAtherosclerosis +11

Design and Synthesis of New Linear and Cyclic Bradykinin Antagonists

Christophe Thurieau, Michel Félétou, Philippe Hennig, +3

Journal of Medicinal Chemistry