Peter A. P. M. van Doremalen

Synthesis and <i>in Vitro</i> and <i>in Vivo</i> Characteristics of an Iodinated Analogue of the β-Adrenoceptor Antagonist Carazolol

Eric A. Dubois, Jan C. Van den Bos, T. Doornbos et al. · Journal of Medicinal Chemistry · 1996 · 32 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +15

The stereoisomers of 17α-[123I]iodovinyloestradiol and its 11α-methoxy derivative evaluated for their oestrogen receptor binding in human MCF-7 cells and rat uterus, and their distribution in immature rats

Leonie J.M. Rijks, Gerard J. Boer, Erik Endert et al. · European Journal of Nuclear Medicine and Molecular Imaging · 1996 · 28 citations

Medicine, Endocrinology, Pharmacology +9

New iodinated progestins as potential ligands for progesterone receptor imaging in breast cancer. part 2: in vivo pharmacological characterization

Leonie J.M. Rijks, Jan C. Van den Bos, Peter A. P. M. van Doremalen et al. · Nuclear Medicine and Biology · 1998 · 15 citations

Medicine, Medicinal Chemistry, Oncology +17

A simple and high‐yield synthesis of (S)‐BZM, (R)‐BZM AND (S)‐IBZM for the preparation of (S)‐¹²³I‐IBZM

M. Bobeldijk, N. P. L. G. Verhoeff, J.A.J.M. Vekemans et al. · Journal of Labelled Compounds and Radiopharmaceuticals · 1990 · 13 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +7

Synthesis, Estrogen Receptor Binding, and Tissue Distribution of a New Iodovinylestradiol Derivative (17α,20E)-21-[123I]Iodo-11β-Nitrato-19-Norpregna-1,3,5(10),20-Tetraene-3,17-Diol (E-[123I]NIVE)

Leonie J.M. Rijks, Jan C. Van den Bos, Peter A. P. M. van Doremalen et al. · Nuclear Medicine and Biology · 1998 · 11 citations

Life Sciences, Endocrinology, Pharmacology +14