R. Scott Lokey

Synthetic molecules that fold into a pleated secondary structure in solution

R. Scott Lokey, Brent L. Iverson · Nature · 1995 · 535 citations

Supramolecular Assembly, Engineering, Natural Sciences +7

Retrospective analysis of natural products provides insights for future discovery trends

Cameron R. Pye, Matthew J. Bertin, R. Scott Lokey et al. · Proceedings of the National Academy of Sciences · 2017 · 529 citations · Full text

Testing the Conformational Hypothesis of Passive Membrane Permeability Using Synthetic Cyclic Peptide Diastereomers

Taha Rezai, Bin Yu, Glenn L. Millhauser et al. · Journal of the American Chemical Society · 2006 · 475 citations

Conformational Flexibility, Internal Hydrogen Bonding, and Passive Membrane Permeability:  Successful in Silico Prediction of the Relative Permeabilities of Cyclic Peptides

Taha Rezai, Jonathan Bock, Mai V. Zhou et al. · Journal of the American Chemical Society · 2006 · 409 citations

Membrane Structure, Proteinlipid Interaction, Biochemistry +12

On-resin N-methylation of cyclic peptides for discovery of orally bioavailable scaffolds

Tina R. White, Chad M. Renzelman, Arthur C Rand et al. · Nature Chemical Biology · 2011 · 373 citations

Medicinal Chemistry, Biochemistry, Natural Sciences +7