Andrei Leitão

In vivo effects of a GPR30 antagonist

Megan K. Dennis, Ritwik Burai, Chinnasamy Ramesh et al. · Nature Chemical Biology · 2009 · 514 citations · Full text

Functional Selectivity, Medicine, Pharmacological Agent +5

Molecular Design, Synthesis and Trypanocidal Activity of Dipeptidyl Nitriles as Cruzain Inhibitors

Leandro A. Alves Avelar, Cristian D. Camilo, Sérgio de Albuquerque et al. · PLoS neglected tropical diseases · 2015 · 81 citations · Full text

Combinatorial Chemistry, Drug Target, Chemical Biology +19

Novel derivatives of 1,3,4-oxadiazoles are potent mitostatic agents featuring strong microtubule depolymerizing activity in the sea urchin embryo and cell culture assays

Alex S. Kiselyov, Marina N. Semenova, Natalya B. Chernyshova et al. · European Journal of Medicinal Chemistry · 2010 · 78 citations

Strong Microtubule, Derivatives, Medicine +8

Characterization, solubility and biological activity of amphihilic biopolymeric Schiff bases synthesized using chitosans

Hellen Franciane Gonçalves Barbosa, Maha Attjioui, Andrei Leitão et al. · Carbohydrate Polymers · 2019 · 69 citations

Biological Activity, Bio-based Nanomaterials, Polysaccharide +2

Exemestane's 17-hydroxylated metabolite exerts biological effects as an androgen

Eric A. Ariazi, Andrei Leitão, Tudor I. Oprea et al. · Molecular Cancer Therapeutics · 2007 · 66 citations

Androgen Receptor, Aromatase Inhibitors, Breast Oncology +10