Wojciech Pietruś

Hydrogen Bonds with Fluorine in Ligand–Protein Complexes-the PDB Analysis and Energy Calculations

Wojciech Pietruś, Rafał Kafel, Andrzej J. Bojarski et al. · Molecules · 2022 · 46 citations · Full text

Natural Sciences, Chemistry, Medicinal Chemistry +16

Dual 5-HT₆ and D₃ Receptor Antagonists in a Group of 1<i>H</i>-Pyrrolo[3,2-<i>c</i>]quinolines with Neuroprotective and Procognitive Activity

Katarzyna Grychowska, Séverine Chaumont‐Dubel, Rafał Kurczab et al. · ACS Chemical Neuroscience · 2019 · 32 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Tuning the activity of known drugs via the introduction of halogen atoms, a case study of SERT ligands – Fluoxetine and fluvoxamine

Jakub Staroń, Wojciech Pietruś, Ryszard Bugno et al. · European Journal of Medicinal Chemistry · 2021 · 32 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

2-Aminoimidazole-based antagonists of the 5-HT6 receptor – A new concept in aminergic GPCR ligand design

Adam S. Hogendorf, Adam S. Hogendorf, Agata Hogendorf et al. · European Journal of Medicinal Chemistry · 2019 · 21 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16

Imidazopyridine-Based 5-HT₆ Receptor Neutral Antagonists: Impact of <i>N</i>¹-Benzyl and <i>N</i>¹-Phenylsulfonyl Fragments on Different Receptor Conformational States

David Vanda, Vittorio Canale, Séverine Chaumont‐Dubel et al. · Journal of Medicinal Chemistry · 2021 · 21 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17