Simon T. Ingate

Synthesis and anti-HIV activity of 1,1,3-trioxo-2H,4H-thieno[3,4-e][1,2,4]thiadiazines (TTDs): a new family of HIV-1 specific non-nucleoside reverse transcriptase inhibitors

Ma Esther Arranz, Simon T. Ingate, Myriam Witvrouw et al. · Bioorganic & Medicinal Chemistry · 1999 · 57 citations

Pharmacy, Medicinal Chemistry, Pharmacology +14

The CSIC [Carbanion mediated Sulfonate (Sulfonamido) Intramolecular Cyclization] reaction: Scope and limitations

JoséL Marco, Simon T. Ingate, Pilar M. Chinchón · Tetrahedron · 1999 · 55 citations

Natural Sciences, Chemistry, Catalysis +1

The CSIC Reaction on Substrates Derived From Aldehydes

José L. Marco, Simon T. Ingate, Carlos Jaime et al. · Tetrahedron · 2000 · 48 citations

Natural Sciences, Chemistry, Biocatalysis +11

1,1,3-Trioxo-2 <i>H</i> ,4 <i>H</i> -Thieno[3,4- <i>e</i> ][1,2,4]Thiadiazine (TTD) Derivatives: a New Class of Nonnucleoside Human Immunodeficiency Virus Type 1 (HIV-1) Reverse Transcriptase Inhibitors with Anti-HIV-1 Activity

Myriam Witvrouw, María Esther Arranz, Christophe Pannecouque et al. · Antimicrobial Agents and Chemotherapy · 1998 · 42 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Studies into the synthesis of derivatives of 4-amino-2,3-dihydroisothiazole 1,1-dioxides and 4-amino-1,2-oxathiole 2,2-dioxides: The search for linked π-system containing analogues as potential inhibitors of HIV-1 reverse transcriptase

Simon T. Ingate, JoséL Marco, Myriam Witvrouw et al. · Tetrahedron · 1997 · 39 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +13