Kyungbo Kim

Impact of linker length on the activity of PROTACs

Kedra Cyrus, Marie Wehenkel, Eunyoung Choi et al. · Molecular BioSystems · 2010 · 223 citations · Full text

Molecular Regulation, Estrogen Receptor, Molecular Biology +23

LMP2-Specific Inhibitors: Chemical Genetic Tools for Proteasome Biology

Yik Khuan Ho, Paola Bargagna‐Mohan, Marie Wehenkel et al. · Chemistry & Biology · 2007 · 114 citations · Full text

Protein Function, Natural Sciences, Lmp2-specific Inhibitors +3

Structure-Based Design of β1i or β5i Specific Inhibitors of Human Immunoproteasomes

Gerjan de Bruin, E.M. Huber, Bo‐Tao Xin et al. · Journal of Medicinal Chemistry · 2014 · 97 citations · Full text

Proteasome Inhibitors, Drug Target, Human Immunoproteasomes +23

Targeted Degradation of the Aryl Hydrocarbon Receptor by the PROTAC Approach: A Useful Chemical Genetic Tool

Hyosung Lee, Dinesh Puppala, Eun‐Young Choi et al. · ChemBioChem · 2007 · 93 citations

Bioorganic Chemistry, Molecular Biology, Chemical Biology +18

Jostling for Position: Optimizing Linker Location in the Design of Estrogen Receptor‐Targeting PROTACs

Kedra Cyrus, Marie Wehenkel, Eun‐Young Choi et al. · ChemMedChem · 2010 · 90 citations

Breast Oncology, Engineering, Chemoprevention Strategy +22