Moses Moustakim

Discovery of an MLLT1/3 YEATS Domain Chemical Probe

Moses Moustakim, Thomas Christott, Octovia Monteiro et al. · Angewandte Chemie International Edition · 2018 · 91 citations · Full text

Molecular Biology, Chemistry, Cancer Biology +18

Discovery of a PCAF Bromodomain Chemical Probe

Moses Moustakim, Peter G. K. Clark, Laura Trulli et al. · Angewandte Chemie International Edition · 2016 · 87 citations · Full text

Structure-Based Approach toward Identification of Inhibitory Fragments for Eleven-Nineteen-Leukemia Protein (ENL)

David Heidenreich, Moses Moustakim, Jurema Schmidt et al. · Journal of Medicinal Chemistry · 2018 · 41 citations · Full text

Structural Bioinformatics, Biomolecular Structure Prediction, Molecular Biology +20

Structural Insights into Interaction Mechanisms of Alternative Piperazine-urea YEATS Domain Binders in MLLT1

Xiaomin Ni, David Heidenreich, Thomas Christott et al. · ACS Medicinal Chemistry Letters · 2019 · 31 citations · Full text

Drug Target, Protein Assembly, Molecular Biology +22

Discovery of a novel allosteric inhibitor scaffold for polyadenosine-diphosphate-ribose polymerase 14 (PARP14) macrodomain 2

Moses Moustakim, Kerstin Riedel, M. Schuller et al. · Bioorganic & Medicinal Chemistry · 2018 · 30 citations · Full text

Medicinal Chemistry, Pharmaceutical Chemistry, Bioorganic Chemistry +15