Paul R. Werkhoven

Peptido Sulfonyl Fluorides as New Powerful Proteasome Inhibitors

Arwin J. Brouwer, Anika M. Jonker, Paul R. Werkhoven et al. · Journal of Medicinal Chemistry · 2012 · 73 citations

Pharmacy, Medicinal Chemistry, Pharmacology +10

Broad-Spectrum Antimalarial Activity of Peptido Sulfonyl Fluorides, a New Class of Proteasome Inhibitors

Serena Tschan, Arwin J. Brouwer, Paul R. Werkhoven et al. · Antimicrobial Agents and Chemotherapy · 2013 · 35 citations · Full text

Medicine, Infectious Diseases, Pharmacology +15

Versatile convergent synthesis of a three peptide loop containing protein mimic of whooping cough pertactin by successive Cu(I)‐catalyzed azide alkyne cycloaddition on an orthogonal alkyne functionalized TAC‐scaffold

Paul R. Werkhoven, Helmus van de Langemheen, Steffen van der Wal et al. · Journal of Peptide Science · 2014 · 29 citations

Life Sciences, Medicinal Chemistry, Molecular Biology +14

Molecular construction of HIV-gp120 discontinuous epitope mimics by assembly of cyclic peptides on an orthogonal alkyne functionalized TAC-scaffold

Paul R. Werkhoven, Mohèb Elwakiel, Theodorus J. Meuleman et al. · Organic & Biomolecular Chemistry · 2015 · 18 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +17