Localization and pharmacological characterization of high affinity binding sites for vasopressin and oxytocin in the rat brain by light microscopic autoradiography

E. Tribollet, Claude Barberis, Serge Jard, +2

Brain Research

Pharmacological CharacterizationRat BrainLight Microscopic AutoradiographyNeuroendocrine MechanismNeurochemistry +14

Vasopressin antagonists allow demonstration of a novel type of vasopressin receptor in the rat adenohypophysis.

Serge Jard, Rolf C. Gaillard, Gilles Guillon, +5

Molecular Pharmacology

The Binding Site of Neuropeptide Vasopressin V1a Receptor

Bernard Mouillac, Bice Chini, Marie‐Noëlle Balestre, +6

Journal of Biological Chemistry

Avp-binding SiteReceptor Functional DomainsMolecular BiologyBinding SiteHypothalamic Peptide +16

Characterization of SR 121463A, a highly potent and selective, orally active vasopressin V2 receptor antagonist.

C. Serradeil‐Le Gal, C Lacour, G Valette, +17

Journal of Clinical Investigation

Molecular PharmacologySelective AffinityArginine VasopressinSr 121463AFunctional Selectivity +12

Angiotensin II and dopamine modulate both cAMP and inositol phosphate productions in anterior pituitary cells. Involvement in prolactin secretion.

A Enjalbert, Fritz Sladeczek, Gilles Guillon, +7

Journal of Biological Chemistry

Cellular PhysiologyGastrointestinal Peptide HormoneAnterior Pituitary CellsMolecular PharmacologyPituitary Gland +15

125I-labelled d(CH2)5[Tyr(Me)2,Thr4,Tyr-NH29]OVT: a selective oxytocin receptor ligand

Jack Elands, Claude Barberis, Serge Jard, +5

European Journal of Pharmacology

Functional SelectivityMedicine125I-labelled DMolecular BiologyMechanism Of Action +3

Specific Binding of [3H]Lysine-Vasopressin to Pig Kidney Plasma Membranes

Joël Bockaert, Christian Roy, Rabary M. Rajerison, +1

Journal of Biological Chemistry

Pig Kidney MedullaExperimental PharmacologyPlasma Membrane FractionCellular PhysiologyMembrane Preparation +15

Angiotensin II and alpha-adrenergic agonists inhibit rat liver adenylate cyclase.

Serge Jard, B. Cantau, K H Jakobs

Journal of Biological Chemistry

HypertensionCardiovascular PharmacologyCellular PharmacologyPharmacotherapyMm Edta +14

Tyr115 is the key residue for determining agonist selectivity in the V1a vasopressin receptor.

Bice Chini, Bernard Mouillac, M N Balestre, +6

The EMBO Journal

Molecular PharmacologySignal TransductionMolecular PhysiologyAgonist SelectivityG Protein-coupled Receptor +11

Oxytocin-sensitive Adenylate Cyclase in Frog Bladder Epithelial Cells

Joël Bockaert, Christian Roy, Serge Jard

Journal of Biological Chemistry

Cellular PharmacologyCytoskeletonEthylene Glycol BisExperimental PharmacologyCellular Physiology +19