Greg Delahanty

Design, Synthesis, and Pharmacological Evaluation of Bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl Sulfide 3 (BPTES) Analogs as Glutaminase Inhibitors

Krupa H. Shukla, Dana Ferraris, Ajit G. Thomas et al. · Journal of Medicinal Chemistry · 2012 · 192 citations · Full text

Pharmaceutical Science, Glutaminase Inhibitors, Pharmacotherapy +16

Synthesis and Biological Evaluation of Thiol-Based Inhibitors of Glutamate Carboxypeptidase II:  Discovery of an Orally Active GCP II Inhibitor

Pavel Majer, Paul Jackson, Greg Delahanty et al. · Journal of Medicinal Chemistry · 2003 · 106 citations · Full text

Molecular Pain, Pharmacotherapy, Chemical Biology +20

Design, Synthesis, and Pharmacological Evaluation of Fluorinated Tetrahydrouridine Derivatives as Inhibitors of Cytidine Deaminase

Dana Ferraris, Bridget Duvall, Greg Delahanty et al. · Journal of Medicinal Chemistry · 2014 · 54 citations · Full text

Cda Substrate, Medicinal Chemistry, Cda-mediated Metabolism +15

Structural Optimization of Thiol-Based Inhibitors of Glutamate Carboxypeptidase II by Modification of the P1‘ Side Chain

Pavel Majer, Bunda Hin, Doris Stoermer et al. · Journal of Medicinal Chemistry · 2006 · 40 citations · Full text

Design, Synthesis, and Pharmacological Evaluation of Glutamate Carboxypeptidase II (GCPII) Inhibitors Based on Thioalkylbenzoic Acid Scaffolds

Doris Stoermer, Dilrukshi Vitharana, Niyada Hin et al. · Journal of Medicinal Chemistry · 2012 · 27 citations · Full text

Molecular Pain, Pharmacotherapy, Pharmaceutical Chemistry +20