Kartik Keertikar

Discovery of pyrazolo[1,5-a]pyrimidine-based CHK1 inhibitors: A template-based approach—Part 2

Marc Labroli, Kamil Paruch, Michael P. Dwyer et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 74 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Drug Target +9

The application of disubstituted vinylogous iminium salts and related synthons to the regiocontrolled preparation of unsymmetrical 2,3,4-trisubstituted pyrroles

John T. Gupton, Keith E. Krumpe, Bruce S. Burnham et al. · Tetrahedron · 1998 · 50 citations

Enantioselective Synthesis, Unsymmetrical 2,3,4-Trisubstituted Pyrroles, Engineering +7

Design and Synthesis of Piperazine Sulfonamide Cores Leading to Highly Potent HIV-1 Protease Inhibitors

Christopher J. Bungard, Peter Williams, Jürgen Schulz et al. · ACS Medicinal Chemistry Letters · 2017 · 43 citations · Full text

Discovery of pyrazolo[1,5-a]pyrimidine-based Pim inhibitors: A template-based approach

Michael P. Dwyer, Kartik Keertikar, Kamil Paruch et al. · Bioorganic & Medicinal Chemistry Letters · 2013 · 40 citations · Full text

Medicinal Chemistry, Medicine, Rational Drug Design +5

The application of vinylogous iminium salt derivatives to an efficient synthesis of the pyrrole containing alkaloids Rigidin and Rigidin E

John T. Gupton, Edith J. Banner, Austin B. Scharf et al. · Tetrahedron · 2006 · 37 citations

Bioorganic Chemistry, Alkaloids Rigidin, Natural Sciences +9