Synthesis and Pharmacological Evaluation of 2,4-Dinitroaryldithiocarbamate Derivatives as Novel Monoacylglycerol Lipase Inhibitors

Coco N. Kapanda, Julien Masquelier, Geoffray Labar, +3

Journal of Medicinal Chemistry

Bis(dialkylaminethiocarbonyl)disulfides as Potent and Selective Monoglyceride Lipase Inhibitors

Coco N. Kapanda, Giulio G. Muccioli, Geoffray Labar, +2

Journal of Medicinal Chemistry

Medicinal ChemistryLipid SynthesisBiochemistryNatural SciencesMedicine +6

Effects of nalfurafine on the reinforcing, thermal antinociceptive, and respiratory-depressant effects of oxycodone: modeling an abuse-deterrent opioid analgesic in rats

E. Andrew Townsend, Jennifer E. Naylor, S. Stevens Negus, +10

Psychopharmacology

Abuse-deterrent Opioid AnalgesicPain MedicineAddictionPhysiologyMedicine +10

Molecular Identification of N-Acetylaspartylglutamate Synthase and β-Citrylglutamate Synthase

François Collard, Vincent Stroobant, Pedro Lamosa, +6

Journal of Biological Chemistry

BiosynthesisProtein ExpressionCellular EnzymologyBiochemistryNatural Sciences +10

PET imaging of fatty acid amide hydrolase in the brain: synthesis and biological evaluation of an 11C-labelled URB597 analogue

Leonie Wyffels, Giulio G. Muccioli, Coco N. Kapanda, +4

Nuclear Medicine and Biology

Positron Emission TomographyBiochemistryPet ImagingMagnetic Resonance SpectroscopyPet-mri +7

Synthesis and pharmacological evaluation of antioxidant chalcone derivatives of 2(3H)-benzoxazolones

Hocine Aichaoui, Faouzi Guenadil, Coco N. Kapanda, +3

Medicinal Chemistry Research

Pharmaceutical ChemistryMedicineOrganic ChemistryHeterocycle ChemistryPharmacology +2

Search for monoglyceride lipase inhibitors: synthesis and screening of arylthioamides derivatives

Coco N. Kapanda, Giulio G. Muccioli, Geoffray Labar, +3

Medicinal Chemistry Research

DerivativesBiochemistryMedicineMonoglyceride Lipase InhibitorsDrug Development +5

<b>Analysis and fragmentation mechanisms of hirsutinolide‐type sesquiterpene lactones by ultra‐high‐performance liquid chromatography/electrospray ionization linear ion trap Orbitrap mass spectrometry</b>

C. Girardi, Valérie Jullian, Mohamed Haddad, +6

Rapid Communications in Mass Spectrometry

EngineeringBiological Mass SpectrometryFragmentation PathwaysBioanalysisAnalytical Chemistry +15