Kasia Kieltyka

A high‐throughput bioanalytical platform using automated infusion for tandem mass spectrometric method optimization and its application in a metabolic stability screen

Kasia Kieltyka, Jun Zhang, Li Shu et al. · Rapid Communications in Mass Spectrometry · 2009 · 52 citations

Pharmacy, Biochemistry, Pharmacology +13

Discovery of 3-hydroxy-4-cyano-isoquinolines as novel, potent, and selective inhibitors of human 11β-hydroxydehydrogenase 1 (11β-HSD1)

Shung Wu, David Yoon, Janice E. Chin et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 28 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +9

Potent Long-Acting Inhibitors Targeting the HIV-1 Capsid Based on a Versatile Quinazolin-4-one Scaffold

Eric P. Gillis, Michael Bowsher, James H. Cook et al. · Journal of Medicinal Chemistry · 2023 · 24 citations

Pharmacy, Pharmacokinetics, Pharmacology +17

An integrated bioanalytical platform for supporting high‐throughput serum protein binding screening

Jun Zhang, Wilson Z. Shou, Marianne Vath et al. · Rapid Communications in Mass Spectrometry · 2010 · 23 citations

Pharmacy, Biochemistry, Medicinal Chemistry +16

Application of Cassette Ultracentrifugation Using Non-labeled Compounds and Liquid Chromatography-Tandem Mass Spectrometry Analysis for High-Throughput Protein Binding Determination

Kasia Kieltyka, Brian McAuliffe, Christopher Cianci et al. · Journal of Pharmaceutical Sciences · 2016 · 15 citations

Life Sciences, Biochemistry, Molecular Biology +16