Jiangkun Yan

Design, synthesis and biological evaluation of tetrahydroquinoline-based reversible LSD1 inhibitors

Xinran Wang, Cai Zhang, Xiangyu Zhang et al. · European Journal of Medicinal Chemistry · 2020 · 37 citations · Full text

Combinatorial Chemistry, Medicinal Chemistry, Biochemistry +7

Design, synthesis and biological evaluation of novel benzofuran derivatives as potent LSD1 inhibitors

Xiangyu Zhang, Hai‐Lan Huang, Ziheng Zhang et al. · European Journal of Medicinal Chemistry · 2021 · 36 citations · Full text

Medicinal Chemistry, Biochemistry, Medicine +11

Molecular docking, 3D-QSAR, and molecular dynamics simulations of thieno[3,2-b]pyrrole derivatives against anticancer targets of KDM1A/LSD1

Xiangyu Zhang, Jiangkun Yan, Hanxun Wang et al. · Journal of Biomolecular Structure and Dynamics · 2020 · 30 citations

Design, synthesis and biological evaluation of curcumin analogues as novel LSD1 inhibitors

Jiming Wang, Xiangyu Zhang, Jiangkun Yan et al. · Bioorganic & Medicinal Chemistry Letters · 2019 · 25 citations · Full text

Medicinal Chemistry, Pharmaceutical Chemistry, Biochemistry +11

Diversity-oriented synthesis and bioactivity evaluation of N-substituted ferrocifen compounds as novel antiproliferative agents against TNBC cancer cells

Yong Wang, Pascal Pigeon, Wei Li et al. · European Journal of Medicinal Chemistry · 2022 · 23 citations · Full text

Diversity Oriented Synthesis, Medicine, Diversity-oriented Synthesis +6