Jean‐Robert Labrosse

Discovery of (2<i>S</i>)-8-[(3<i>R</i>)-3-Methylmorpholin-4-yl]-1-(3-methyl-2-oxobutyl)-2-(trifluoromethyl)-3,4-dihydro-2<i>H</i>-pyrimido[1,2-<i>a</i>]pyrimidin-6-one: A Novel Potent and Selective Inhibitor of Vps34 for the Treatment of Solid Tumors

Benoit Pasquier, Youssef El‐Ahmad, Bruno Filoche-Rommé et al. · Journal of Medicinal Chemistry · 2014 · 90 citations

Drug Target, Solid Tumors, Exquisite Selectivity +22

Chiral Aromatase and Dual Aromatase−Steroid Sulfatase Inhibitors from the Letrozole Template: Synthesis, Absolute Configuration, and In Vitro Activity

Paul M. Wood, L. W. Lawrence Woo, Jean‐Robert Labrosse et al. · Journal of Medicinal Chemistry · 2008 · 85 citations · Full text

A Simple and Efficient Enantioselective Synthesis of 2-Alkylidene-3-alkyl-1,4-benzodioxanes by Palladium-Catalyzed Annulation of Benzene-1,2-diol and Propargylic Carbonates

Jean‐Robert Labrosse, Paul Lhoste, Denis Sinou · Organic Letters · 2000 · 65 citations

Various Propargylic Carbonates, Engineering, Chiral Atropoisomeric Diphosphine +12

An easy palladium-catalyzed access to 2-alkylidene-1,4-benzodioxanes

Jean‐Robert Labrosse, Paul Lhoste, Denis Sinou · Tetrahedron Letters · 1999 · 64 citations

Easy Palladium-catalyzed Access, Engineering, Organic Chemistry +4

Palladium-Catalyzed Synthesis of 2,3-Dihydro-2-ylidene-1,4-benzodioxins

Jean‐Robert Labrosse, Paul Lhoste, Denis Sinou · The Journal of Organic Chemistry · 2001 · 53 citations