Léopold Thabault

1-(2-Hydroxybenzoyl)-thiosemicarbazides are promising antimicrobial agents targeting d-alanine-d-alanine ligase in bacterio

Alice Ameryckx, Léopold Thabault, Lionel Pochet et al. · European Journal of Medicinal Chemistry · 2018 · 34 citations · Full text

Antimicrobial Drug Discovery, D-alanine-d-alanine Ligase, Medicine +8

Olaparib Is a Mitochondrial Complex I Inhibitor That Kills Temozolomide-Resistant Human Glioblastoma Cells

Luca X. Zampieri, Martina Sboarina, Andrea Cacace et al. · International Journal of Molecular Sciences · 2021 · 27 citations · Full text

Parp Inhibitor Olaparib, Dna Repair Inhibition, High-grade Gliomas +16

Interrogating the Lactate Dehydrogenase Tetramerization Site Using (Stapled) Peptides

Léopold Thabault, Lucie Brisson, Chiara Brustenga et al. · Journal of Medicinal Chemistry · 2020 · 23 citations · Full text

Protein Assembly, Peptide Engineering, Lactate Dehydrogenases +16

Discovery of a novel lactate dehydrogenase tetramerization domain using epitope mapping and peptides

Léopold Thabault, Maxime Liberelle, Katarina Koruza et al. · Journal of Biological Chemistry · 2021 · 17 citations · Full text

Rational Design of Original Fused-Cycle Selective Inhibitors of Tryptophan 2,3-Dioxygenase

Arina Kozlova, Léopold Thabault, Maxime Liberelle et al. · Journal of Medicinal Chemistry · 2021 · 17 citations · Full text