G Protein-Coupled Receptor 30 Localizes to the Endoplasmic Reticulum and Is Not Activated by Estradiol

Christiane Otto, Beate Rohde-Schulz, Gilda Schwarz, +8

Endocrinology

Classical Estrogen ReceptorEstradiol StimulationCellular PhysiologyMolecular PharmacologyEndocytic Pathway +15

The plasminogen activator family from the salivary gland of the vampire bat Desmodus rotundas: cloning and expression

Jörn Krätzschmar, Bernard Haendler, Gernot Langer, +5

Gene

BiologyPlasminogen Activator FamilyNatural SciencesPathogenesisOral Biology +6

The Cochaperone Bag-1L Enhances Androgen Receptor Action via Interaction with the NH₂-Terminal Region of the Receptor

Liubov Shatkina, Sigrun Mink, Hermann Rogatsch, +4

Molecular and Cellular Biology

Androgen ReceptorTau 5Molecular BiologyMolecular Chaperone Hsp70Molecular Pharmacology +15

Plasmhogen Activators from the Saliva of <i>Desmodus rotundus</i> (Common Vampire Bat): Unique Fibrin Specificity

Wolf‐Dieter Schleuning, Alejandro Alagón, Werner Boidol, +8

Annals of the New York Academy of Sciences

GeneticsMolecular BiologySingle Chain TpaMolecular GeneticsSalivary Gland +20

Structural Evidence for Isoform-Selective Allosteric Inhibition of Lactate Dehydrogenase A

Anders Friberg, Hartmut Rehwinkel, Duy Nguyen, +6

ACS Omega

Medicinal ChemistryBiosynthesisAldehyde DehydrogenaseBiochemistryStructural Evidence +10

Discovery of BAY-298 and BAY-899: Tetrahydro-1,6-naphthyridine-Based, Potent, and Selective Antagonists of the Luteinizing Hormone Receptor Which Reduce Sex Hormone Levels in Vivo

Lars Wortmann, B. Lindenthal, Peter Muhn, +17

Journal of Medicinal Chemistry

Sex HormonesGynecologyPharmacotherapyPharmaceutical ChemistryMedicinal Chemistry +15

Production of vampire bat plasminogen activator DSPA α1 in CHO and insect cells

Thomas Petri, Gernot Langer, Peter Bringmann, +4

Journal of Biotechnology

BiologyInsect CellsNatural SciencesGene ExpressionMedicine +3

Identification of a Benzimidazolecarboxylic Acid Derivative (<b>BAY 1316957</b>) as a Potent and Selective Human Prostaglandin E2 Receptor Subtype 4 (hEP4-R) Antagonist for the Treatment of Endometriosis

Stefan Bäurle, Jens Nagel, Olaf Peters, +11

Journal of Medicinal Chemistry

Pain MedicineGynecologyMolecular PainPharmacotherapyPharmaceutical Chemistry +14

Synthesis and biological activities of a new series of secosteroids: vitamin D phosphonate hybrids

Andreas Steinmeyer, Katica Schwarz, Martin Haberey, +2

Steroids

BiosynthesisBiochemistryNatural SciencesDiversity-oriented SynthesisNatural Product Biosynthesis +5

Discovery and Characterization of BAY 1214784, an Orally Available Spiroindoline Derivative Acting as a Potent and Selective Antagonist of the Human Gonadotropin-Releasing Hormone Receptor as Proven in a First-In-Human Study in Postmenopausal Women

Olaf Panknin, Andrea Wagenfeld, Wilhelm Bone, +14

Journal of Medicinal Chemistry