Jesús García

New peptide architectures through C–H activation stapling between tryptophan–phenylalanine/tyrosine residues

Lorena Mendive‐Tapia, Sara Preciado, Jesús García et al. · Nature Communications · 2015 · 296 citations · Full text

Pharmacy, Biochemistry, Medicinal Chemistry +17

Synthesis of Ecteinascidin ET-743 and Phthalascidin Pt-650 from Cyanosafracin B

Carmen Cuevas, Marta del Pozo Pérez, María Jesús Martín et al. · Organic Letters · 2000 · 281 citations

Natural Sciences, Chemistry, Organic Chemistry +1

Small molecule inhibits α-synuclein aggregation, disrupts amyloid fibrils, and prevents degeneration of dopaminergic neurons

Jordi Pujols, Samuel Peña‐Díaz, Diana F. Lázaro et al. · Proceedings of the National Academy of Sciences · 2018 · 233 citations · Full text

Life Sciences, Neurobiology, Neuroscience +17

Stapled Peptides by Late‐Stage C(sp³)−H Activation

Anaïs F. M. Noisier, Jesús García, Ioana Ionuț et al. · Angewandte Chemie International Edition · 2016 · 160 citations

Pharmacy, Biochemistry, Medicinal Chemistry +13

EPI-001, A Compound Active against Castration-Resistant Prostate Cancer, Targets Transactivation Unit 5 of the Androgen Receptor

Eva De Mol, R. Bryn Fenwick, Christopher T. W. Phang et al. · ACS Chemical Biology · 2016 · 156 citations · Full text

Medicine, Medicinal Chemistry, Oncology +17