Concepedia
Statistics
Publications
3
Citations
137
H-Index
Active since
2017
Affiliations
Inserm(Current)
Université de Lille
Université de Montpellier
Centre de Recherche Jean Pierre Aubert
Centre de Biologie Structurale
Floriane Gibault is an author at Inserm specializing in drug development, drug discovery, and medicinal chemistry.
Top concepts
MedicineBiochemistryPharmacologyDrug DiscoveryDrug DevelopmentNatural SciencesMedicinal ChemistryBiomolecular Engineering
Publications per year
2017–2021
Molecular Features of the YAP Inhibitor Verteporfin: Synthesis of Hexasubstituted Dipyrrins as Potential Inhibitors of YAP/TAZ, the Downstream Effectors of the Hippo Pathway
Floriane Gibault, Fabrice Bailly, Matthieu Corvaisier et al. · ChemMedChem · 2017 · 76 citations · Full text
Toward the Discovery of a Novel Class of YAP–TEAD Interaction Inhibitors by Virtual Screening Approach Targeting YAP–TEAD Protein–Protein Interface
Floriane Gibault, Mathilde Coevoet, Manon Sturbaut et al. · Cancers · 2018 · 43 citations · Full text
Design, Synthesis and Evaluation of a Series of 1,5‐Diaryl‐1,2,3‐triazole‐4‐carbohydrazones as Inhibitors of the YAP‐TAZ/TEAD Complex
Floriane Gibault, Manon Sturbaut, Mathilde Coevoet et al. · ChemMedChem · 2021 · 18 citations
Medicinal Chemistry, Yap-tead Interaction, Biochemistry +13
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