Aldrin V. Vasco

Macrocyclization of Peptide Side Chains by the Ugi Reaction: Achieving Peptide Folding and Exocyclic <i>N</i>-Functionalization in One Shot

Aldrin V. Vasco, Carlos Pérez, Fidel E. Morales et al. · The Journal of Organic Chemistry · 2015 · 60 citations

Life Sciences, Biochemistry, Medicinal Chemistry +17

A Multicomponent Stapling Approach to Exocyclic Functionalized Helical Peptides: Adding Lipids, Sugars, PEGs, Labels, and Handles to the Lactam Bridge

Aldrin V. Vasco, Yanira Méndez, Andrea Porzel et al. · Bioconjugate Chemistry · 2018 · 57 citations

Life Sciences, Biochemistry, Medicinal Chemistry +15

Multicomponent polysaccharide–protein bioconjugation in the development of antibacterial glycoconjugate vaccine candidates

Yanira Méndez, Janoi Chang, Ana R. Humpierre et al. · Chemical Science · 2018 · 53 citations · Full text

Pharmacy, Biotechnology, Immunology +17

Discovery of potent and selective inhibitors of the Escherichia coli M1-aminopeptidase via multicomponent solid-phase synthesis of tetrazole-peptidomimetics

Yanira Méndez, German De Armas, Idalia Pérez et al. · European Journal of Medicinal Chemistry · 2018 · 38 citations

Pharmacy, Biochemistry, Medicinal Chemistry +16

A Multicomponent Conjugation Strategy to Unique <i>N‐</i>Steroidal Peptides: First Evidence of the Steroidal Nucleus as a β‐Turn Inducer in Acyclic Peptides

Daniel G. Rivera, Aldrin V. Vasco, Radell Echemendía et al. · Chemistry - A European Journal · 2014 · 28 citations

Life Sciences, Biochemistry, Medicinal Chemistry +17