Stéphane Bourg

PKIDB: A Curated, Annotated and Updated Database of Protein Kinase Inhibitors in Clinical Trials

Fabrice Carles, Stéphane Bourg, Christophe Meyer et al. · Molecules · 2018 · 182 citations · Full text

Drug Target, Kinase Inhibitors, Pharmacotherapy +26

Synthesis of chromeno[3,4-b]indoles as Lamellarin D analogues : A novel DYRK1A inhibitor class

Cléopatra Neagoie, Emeline Vedrenne, Frédéric Buron et al. · European Journal of Medicinal Chemistry · 2012 · 98 citations · Full text

Medicinal Chemistry, Pharmaceutical Chemistry, Bioorganic Chemistry +9

Design, Synthesis, and Biological Activity of Pyridopyrimidine Scaffolds as Novel PI3K/mTOR Dual Inhibitors

Thibault Saurat, Frédéric Buron, Nuno F. Rodrigues et al. · Journal of Medicinal Chemistry · 2013 · 83 citations · Full text

Combinatorial Chemistry, Dual Pi3k/mtor Inhibitors, Medicinal Chemistry +16

Comparative Assessment of Protein Kinase Inhibitors in Public Databases and in PKIDB

Colin Bournez, Fabrice Carles, Gautier Peyrat et al. · Molecules · 2020 · 68 citations · Full text

Novel Tetrahydropyrido[1,2-<i>a</i>]isoindolone Derivatives (Valmerins): Potent Cyclin-Dependent Kinase/Glycogen Synthase Kinase 3 Inhibitors with Antiproliferative Activities and Antitumor Effects in Human Tumor Xenografts

Rajâa Boulahjar, Aziz Ouach, Matteo Chiurato et al. · Journal of Medicinal Chemistry · 2012 · 53 citations · Full text

Peptide Science, Human Tumor Xenografts, Pharmaceutical Chemistry +19