New non competitive AMPA antagonists

Gizella Ábrahám, Sándor Sólyom, Emese Csuzdi, +12

Bioorganic & Medicinal Chemistry

Functional SelectivityMedicineMechanism Of ActionPharmacotherapyElectrophysiology +3

Antagonism of AMPA receptors produces anxiolytic-like behavior in rodents: Effects of GYKI 52466 and its novel analogues

Gábor Kapus, István Gacsályi, Miklós Végh, +7

Psychopharmacology

Signal TransductionBiochemistryFunctional SelectivityMedicinePhysiology +10

The effects of AMPA receptor antagonists in models of stroke and neurodegeneration

Pierre Gressèns, Michael Spedding, Gábor Gigler, +9

European Journal of Pharmacology

Ischemic StrokeNeurophysiologyStrokeMedicineNeuropharmacology +10

Tianeptine potentiates AMPA receptors by activating CaMKII and PKA via the p38, p42/44 MAPK and JNK pathways

Viktor Szegedi, Gábor Juhász, Xiaoqun Zhang, +7

Neurochemistry International

Molecular PhysiologySignal TransductionBiochemistryG Protein-coupled ReceptorMedicine +11

A novel GABAA alpha 5 receptor inhibitor with therapeutic potential

István Ling, Balázs Mihalik, L.-A. Etherington, +20

European Journal of Pharmacology

Functional SelectivityMedicineDrug DiscoveryG Protein-coupled ReceptorMechanism Of Action +7

AMPA receptor antagonists, GYKI 52466 and NBQX, do not block the induction of long-term potentiation at therapeutically relevant concentrations

Gábor Kapus, József I. Székely, J. Durand, +2

Brain Research Bulletin

Functional SelectivityMedicinePhysiologyGyki 52466Receptor (Biochemistry) +9

Neuroprotective and anticonvulsant effects of EGIS‐8332, a non‐competitive AMPA receptor antagonist, in a range of animal models

Gábor Gigler, Krisztina Móricz, Márta Ágoston, +13

British Journal of Pharmacology

Comparison of the AMPA Antagonist Action of New 2,3-Benzodiazepines in Vitro and Their Neuroprotective Effects in Vivo

Gábor Kapus, Szabolcs Kertész, Gábor Gigler, +5

Pharmaceutical Research

NeurophysiologyNew 2,3-BenzodiazepinesMedicineAnesthetic MechanismTheir Neuroprotective Effects +10

Interactions of allosteric modulators of AMPA/kainate receptors on spreading depression in the chicken retina

Szabolcs Kertész, Gábor Kapus, György Lévay

Brain Research

Allosteric ModulatorsNeurotransmitterNeurotransmissionOptogeneticsGanglion Cell +14

Deramciclane improves object recognition in rats: Potential role of NMDA receptors

Szabolcs Kertész, Gábor Kapus, István Gacsályi, +1

Pharmacology Biochemistry and Behavior

NeurophysiologyNeuroanatomyMedicineNmda ReceptorsNeuropeptide Receptor +8