Fredrik R. Zetterberg

Target inhibition of galectin-3 by inhaled TD139 in patients with idiopathic pulmonary fibrosis

Nikhil Hirani, Alison C. MacKinnon, Lisa Nicol et al. · European Respiratory Journal · 2020 · 205 citations · Full text

An Orally Active Galectin-3 Antagonist Inhibits Lung Adenocarcinoma Growth and Augments Response to PD-L1 Blockade

Lynda Vuong, Eleni Kouverianou, Claire Rooney et al. · Cancer Research · 2019 · 138 citations · Full text

Extracellular and intracellular small-molecule galectin-3 inhibitors

John Stegmayr, Fredrik R. Zetterberg, Michael C. Carlsson et al. · Scientific Reports · 2019 · 104 citations · Full text

Monosaccharide Derivatives with Low‐Nanomolar Lectin Affinity and High Selectivity Based on Combined Fluorine–Amide, Phenyl–Arginine, Sulfur–π, and Halogen Bond Interactions

Fredrik R. Zetterberg, Kristoffer Peterson, Richard Johnsson et al. · ChemMedChem · 2017 · 102 citations

Glycobiology, Organic Chemistry, Peptide Science +23

Systematic Tuning of Fluoro-galectin-3 Interactions Provides Thiodigalactoside Derivatives with Single-Digit nM Affinity and High Selectivity

Kristoffer Peterson, Rohit Kumar, Olof Stenström et al. · Journal of Medicinal Chemistry · 2017 · 98 citations · Full text