Janet E. Rivett

New nonpeptide angiotensin II receptor antagonists. 3. Synthesis, biological properties, and structure-activity relationships of 2-alkyl-4-(biphenylylmethoxy)pyridine derivatives

Robert H. Bradbury, C. Allott, Michael Robert Dennis et al. · Journal of Medicinal Chemistry · 1993 · 70 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +11

1,2,4-Triazolo[4,3-a]pyrazine derivatives with human renin inhibitory activity. 3. Synthesis and biological properties of aminodeoxystatine and difluorostatone derivatives

Robert H. Bradbury, Janet E. Rivett · Journal of Medicinal Chemistry · 1991 · 46 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +9

An efficient synthesis of the γ-lactone corresponding to a hydroxyethylene dipeptide isostere using stereoselective bromolactonisation of a chiral acyloxazolidinone

Robert H. Bradbury, John Revill, Janet E. Rivett et al. · Tetrahedron Letters · 1989 · 28 citations

Natural Sciences, Chemistry, Organic Chemistry +2

1,2,4-Triazolo[4,3-a]pyrazine derivatives with human renin inhibitory activity. 2. Synthesis, biological properties and molecular modeling of hydroxyethylene isostere derivatives

Robert H. Bradbury, John S. Major, Janet E. Rivett et al. · Journal of Medicinal Chemistry · 1990 · 17 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

An Efficient Synthesis of 3-Alkyl-5-aryl-2(1H)-pyrazinones

Robert H. Bradury, Robert H. Bradbury, D. Vaughan Griffiths et al. · Heterocycles · 1990 · 15 citations · Full text

Natural Sciences, Chemistry, Medicinal Chemistry +10