Giacomo Berretta

Inhibitory Kappa B Kinase α (IKKα) Inhibitors That Recapitulate Their Selectivity in Cells against Isoform-Related Biomarkers

Nahoum G. Anthony, Jessica Baiget, Giacomo Berretta et al. · Journal of Medicinal Chemistry · 2017 · 38 citations · Full text

Life Sciences, Cell Biology, Molecular Biology +13

Topographical Mapping of Isoform-Selectivity Determinants for J-Channel-Binding Inhibitors of Sphingosine Kinases 1 and 2

David R. Adams, Salha M. Tawati, Giacomo Berretta et al. · Journal of Medicinal Chemistry · 2019 · 37 citations · Full text

Life Sciences, Biochemistry, Pharmacology +16

Doing the methylene shuffle – Further insights into the inhibition of mitotic kinesin Eg5 with S-trityl l-cysteine

Murad Abualhasan, James A. D. Good, Kitiyaporn Wittayanarakul et al. · European Journal of Medicinal Chemistry · 2012 · 21 citations · Full text

Life Sciences, Cell Biology, Molecular Biology +16

Design and Synthesis of Novel Aminoindazole-pyrrolo[2,3-b]pyridine Inhibitors of IKKα That Selectively Perturb Cellular Non-Canonical NF-κB Signalling

Christopher M. Riley, Usama M. Ammar, Aisha A. Alsfouk et al. · Molecules · 2024 · 12 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +13