Decarbonylative C–H Coupling of Azoles and Aryl Esters: Unprecedented Nickel Catalysis and Application to the Synthesis of Muscoride A

Kazuma Amaike, Kei Muto, Junichiro Yamaguchi, +1

Journal of the American Chemical Society

Chemical EngineeringCross-coupling ReactionEngineeringMuscoride ACatalytic Synthesis +11

β-Selective C–H Arylation of Pyrroles Leading to Concise Syntheses of Lamellarins C and I

Kirika Ueda, Kazuma Amaike, Richard M. Maceiczyk, +2

Journal of the American Chemical Society

β-Selective C–h ArylationEngineeringOrganic ChemistryChemistryHeterocycle Chemistry +14

C7-Derivatization of C3-Alkylindoles Including Tryptophans and Tryptamines

Richard P. Loach, Owen S. Fenton, Kazuma Amaike, +3

The Journal of Organic Chemistry

C3-alkylindoles Including TryptophansChemical EngineeringCross-coupling ReactionEngineeringC7-selective Boronation +9

Affinity-Guided Oxime Chemistry for Selective Protein Acylation in Live Tissue Systems

Tomonori Tamura, Zhining Song, Kazuma Amaike, +4

Journal of the American Chemical Society

Bioorganic ChemistryMolecular BiologyLive Tissue SystemsSelective Protein AcylationEnzymatic Modification +16

Photopharmacological Manipulation of Mammalian CRY1 for Regulation of the Circadian Clock

Dušan Kolarski, Simon Miller, Tsuyoshi Oshima, +12

Journal of the American Chemical Society

Synthesis of Triarylpyridines in Thiopeptide Antibiotics by Using a C−H Arylation/Ring‐Transformation Strategy

Kazuma Amaike, Kenichiro Itami, Junichiro Yamaguchi

Chemistry - A European Journal

Combinatorial ChemistryMedicinal ChemistryEngineeringHeterocyclicC−h Arylation/ring‐transformation Strategy +11

An Isoform-Selective Modulator of Cryptochrome 1 Regulates Circadian Rhythms in Mammals

Simon Miller, Yoshiki Aikawa, Akiko Sugiyama, +7

Cell chemical biology

Signal TransductionAlertnessMedicinePhysiologyIsoform-selective Modulator +10

Synthesis of multiply arylated pyridines

Takashi Asako, Wakana Hayashi, Kazuma Amaike, +4

Tetrahedron

Organic ChemistrySynthetic ChemistrySynthesis MethodChemistry

Late-Stage C–H Coupling Enables Rapid Identification of HDAC Inhibitors: Synthesis and Evaluation of NCH-31 Analogues

Hiromi Sekizawa, Kazuma Amaike, Yukihiro Itoh, +3

ACS Medicinal Chemistry Letters

Potent Pan-hdac InhibitorMolecular PharmacologyMedicinal ChemistryHdac InhibitorsBiochemistry +11

Construction of a Fluorescent Screening System of Allosteric Modulators for the GABA_A Receptor Using a Turn-On Probe

Seiji Sakamoto, Kei Yamaura, Tomohiro Numata, +5

ACS Central Science