Wieslaw Kazmierski

Novel peptidic mu opioid antagonists: pharmacologic characterization in vitro and in vivo.

Thomas H. Kramer, Jennifer E. Shook, Wieslaw Kazmierski et al. · Journal of Pharmacology and Experimental Therapeutics · 1989 · 135 citations

[3H]-[H-D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Pen-Thr-NH2] ([3H]CTOP), a potent and highly selective peptide for mu opioid receptors in rat brain.

Kumiko N. Hawkins, Richard J. Knapp, George K. Lui et al. · Journal of Pharmacology and Experimental Therapeutics · 1989 · 101 citations

A new approach to receptor ligand design: synthesis and conformation of a new class of potent and highly selective μ opioid antagonists utilizing tetrahydroisoouinoline carroxylic acid

Wieslaw Kazmierski, Victor J. Hruby · Tetrahedron · 1988 · 93 citations

Molecular Pharmacology, Diversity Oriented Synthesis, Biochemistry +10

Cholecystokinin analogues with high affinity and selectivity for brain membrane receptors*

Victor J. Hruby, Sunan Fang, Richard J. Knapp et al. · International journal of peptide & protein research · 1990 · 47 citations

Cyclic somatostatin analogues as potent antagonists at μ-, but not δ- and κ-opioid receptors mediating presynaptic inhibition of neurotransmitter release in the brain

Arie H. Mulder, George Wardeh, François Hogenboom et al. · European Journal of Pharmacology · 1991 · 23 citations

Cyclic Somatostatin Analogues, Molecular Pharmacology, Neurophysiology +14