Koen Augustyns

Kinetic Investigation of Chemokine Truncation by CD26/Dipeptidyl Peptidase IV Reveals a Striking Selectivity within the Chemokine Family

Anne‐Marie Lambeir, Paul Proost, Christine Durinx et al. · Journal of Biological Chemistry · 2001 · 275 citations · Full text

Extended Structure–Activity Relationship and Pharmacokinetic Investigation of (4-Quinolinoyl)glycyl-2-cyanopyrrolidine Inhibitors of Fibroblast Activation Protein (FAP)

Koen Jansen, Leen Heirbaut, Robert Verkerk et al. · Journal of Medicinal Chemistry · 2014 · 264 citations · Full text

Structure–activity Relationship, Drug Target, Cellular Pharmacology +17

Selective Inhibitors of Fibroblast Activation Protein (FAP) with a (4-Quinolinoyl)-glycyl-2-cyanopyrrolidine Scaffold

Koen Jansen, Leen Heirbaut, Jonathan D. Cheng et al. · ACS Medicinal Chemistry Letters · 2013 · 246 citations · Full text

Bioorganic Chemistry, Selective Inhibitors, Chemical Biology +17

When PERK inhibitors turn out to be new potent RIPK1 inhibitors: critical issues on the specificity and use of GSK2606414 and GSK2656157

Diego Rojas‐Rivera, Tinneke Delvaeye, Ria Roelandt et al. · Cell Death and Differentiation · 2017 · 193 citations · Full text

Critical Issues, Medicine, Receptor Tyrosine Kinase +7

Fluoro-Olefins as Peptidomimetic Inhibitors of Dipeptidyl Peptidases

Pieter Van der Veken, Kristel Senten, István Kertész et al. · Journal of Medicinal Chemistry · 2004 · 168 citations · Full text

Medicinal Chemistry, Bioorganic Chemistry, Biochemistry +15