Kenneth M. Gigstad - Concepedia

Author

Kenneth M. Gigstad

Millennium Engineering and Integration (United States)

Also Known As

Gigstad, K.M., K. M. GIGSTAD, K. M. Gigstad, Kenneth Gigstad, Kenneth M. Gigstad, Kenneth M. Gigstad

Publications

830

Citations

H-Index

Concepts

All Affiliations

Millennium Engineering and Integration (United States)RTI International Eli Lilly (United States)Purdue University West Lafayette Takeda (United States)

About

Kenneth M. Gigstad is an author at Millennium Engineering and Integration (United States) specializing in biochemistry, natural sciences, and drug discovery.

Top Concepts

#	Concept	H-Index	Publications	Citations
1	Biochemistry	7	7	577
2	Natural Sciences	6	6	560
3	Medicine	5	5	192
4	Chemical Biology	3	3	119
5	Chemistry	3	3	396

Kenneth M. Gigstad

Publications

819

Citations

H-Index

Page 1

	Year	Citations
Asymmetric Catalysis of the Strecker Amino Acid Synthesis by a Cyclic Dipeptide Mani S. Iyer, Kenneth M. Gigstad, Nivedita Namdev, Journal of the American Chemical Society Diversity Oriented SynthesisBiochemistryDonut IconNatural SciencesBiocatalysis	1996	339
Characterization of a new series of non-covalent proteasome inhibitors with exquisite potency and selectivity for the 20S β5-subunit Christopher Blackburn, Kenneth M. Gigstad, Paul Hales, Biochemical Journal	2010	144
N,C-Capped Dipeptides with Selectivity for Mycobacterial Proteasome over Human Proteasomes: Role of S3 and S1 Binding Pockets Gang Lin, Tamutenda Chidawanyika, Christopher Tsu, Journal of the American Chemical Society Protein AssemblyImmunologyMolecular BiologyAntigen ProcessingSpecies Selectivity	2013	56
Asymmetric catalysis of the Strecker amino acid synthesis by a cyclic dipeptide Mani S. Iyer, Kenneth M. Gigstad, Nivedita Namdev, Amino Acids BiochemistryNatural SciencesBiocatalysisEnzyme CatalysisPeptide Synthesis	1996	46
Potent Histone Deacetylase Inhibitors Derived from 4-(Aminomethyl)-<i>N</i>-hydroxybenzamide with High Selectivity for the HDAC6 Isoform Christopher Blackburn, Cynthia Barrett, Janice E. Chin, Journal of Medicinal Chemistry Combinatorial ChemistryHdac6 IsoformChemical BiologyEnzymatic ModificationPharmaceutical Chemistry	2013	42
Identification of Novel Carbocyclic Pyrimidine Cyclic Dinucleotide STING Agonists for Antitumor Immunotherapy Using Systemic Intravenous Route Štěpán Vyskočil, David Cardin, Jeffrey P. Ciavarri, Journal of Medicinal Chemistry	2021	41
Optimization of a series of dipeptides with a P3 threonine residue as non-covalent inhibitors of the chymotrypsin-like activity of the human 20S proteasome Christopher Blackburn, Cynthia Barrett, Jonathan L. Blank, Bioorganic & Medicinal Chemistry Letters Protein ChemistryMedicinal ChemistryP3 Threonine ResidueBiochemistryNatural Sciences	2010	40
Design, Synthesis, and Evaluation of Naphthalene-Sulfonamide Antagonists of Human CCR8 Tracy J. Jenkins, Bing Guan, Mingshi Dai, Journal of Medicinal Chemistry Medicinal ChemistryPharmaceutical ChemistryPharmaceutical ScienceBiochemistryMedicine	2007	37
Discovery of an Opioid κ Receptor Selective Pure Antagonist from a Library of N-Substituted 4β-Methyl-5-(3-hydroxyphenyl)morphans James B. Thomas, Robert N. Atkinson, Nivedita Namdev, Journal of Medicinal Chemistry	2002	29
Histone deacetylase inhibitors derived from 1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine and related heterocycles selective for the HDAC6 isoform Christopher Blackburn, Cynthia Barrett, Mable Brunson, Bioorganic & Medicinal Chemistry Letters BiochemistryMedicineHistone Deacetylase InhibitorsHdac6 IsoformRelated Heterocycles	2014	17

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