Concepedia

Author

Blair T. Lapointe

Merck & Co., Inc., Rahway, NJ, USA (United States)

Also Known As

Blair Lapointe, Blair T. Lapointe, Lapointe, Blair T.

9

Publications

166

Citations

6

H-Index

16

Concepts

All Affiliations

Merck & Co., Inc., Rahway, NJ, USA (United States)
BT

About

Blair T. Lapointe is an author at Merck & Co., Inc., Rahway, NJ, USA (United States) specializing in drug discovery, natural sciences, and drug development.

Top Concepts

#ConceptH-IndexPublicationsCitations

1

Medicine

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88

2

Natural Sciences

2

2

88

3

Biochemistry

2

2

88

4

Biomedical Engineering

1

1

64

5

Biomolecular Engineering

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64

Blair T. Lapointe

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6

Publications

166

Citations

6

H-Index

YearCitations

Strategy for Extending Half-life in Drug Design and Its Significance

Hakan Günaydin, Michael D. Altman, J. Michael Ellis,

ACS Medicinal Chemistry Letters

2018

64

Structure-based design and development of (benz)imidazole pyridones as JAK1-selective kinase inhibitors

Vladimir Simov, Sujal V. Deshmukh, Christopher J. Dinsmore,

Bioorganic & Medicinal Chemistry Letters

2016

24

Discovery of <i>N</i>-(Indazol-3-yl)piperidine-4-carboxylic Acids as RORγt Allosteric Inhibitors for Autoimmune Diseases

Hongjun Zhang, Blair T. Lapointe, Neville J. Anthony,

ACS Medicinal Chemistry Letters

2020

24

Preparation of a Stable Trifluoroborate Salt for the Synthesis of 1-Aryl-2,2-difluoro-enolethers and/or 2,2-Difluoro-1-aryl-ketones via Palladium-Mediated Cross-Coupling

Jason D. Katz, Blair T. Lapointe, Christopher J. Dinsmore

The Journal of Organic Chemistry

2009

21

Discovery and Optimization of Potent, Selective, and Brain-Penetrant 1-Heteroaryl-1 <i>H</i> -Indazole LRRK2 Kinase Inhibitors for the Treatment of Parkinson’s Disease

David A. Candito, Vladimir Simov, Anmol Gulati,

Journal of Medicinal Chemistry

2022

19

Optimization of brain-penetrant picolinamide derived leucine-rich repeat kinase 2 (LRRK2) inhibitors

Anmol Gulati, Charles S. Yeung, Blair T. Lapointe,

RSC Medicinal Chemistry

2021

14

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