Rogelio Siles

Design, synthesis, and biological evaluation of combretastatin nitrogen-containing derivatives as inhibitors of tubulin assembly and vascular disrupting agents

Keith A. Monk, Rogelio Siles, Mallinath B. Hadimani et al. · Bioorganic & Medicinal Chemistry · 2006 · 79 citations

Pharmacy, Medicinal Chemistry, Pharmacology +15

Design, synthesis, and biochemical evaluation of novel cruzain inhibitors with potential application in the treatment of Chagas’ disease

Rogelio Siles, Shen-En Chen, Ming Zhou et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 72 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +6

Combretastatin Dinitrogen-Substituted Stilbene Analogues as Tubulin-Binding and Vascular-Disrupting Agents

Rogelio Siles, J. Freeland Ackley, Mallinath B. Hadimani et al. · Journal of Natural Products · 2008 · 45 citations

Medicine, Medicinal Chemistry, Pharmacology +14

Denatured state aggregation parameters derived from concentration dependence of protein stability

Arne Schön, Benjamin R. Clarkson, Rogelio Siles et al. · Analytical Biochemistry · 2015 · 39 citations

Life Sciences, Biochemistry, Biophysics +15

Development of Synthetic Methodology Suitable for the Radiosynthesis of Combretastatin A-1 (CA1) and Its Corresponding Prodrug CA1P

Anupama Shirali, Madhavi Sriram, John J. Hall et al. · Journal of Natural Products · 2009 · 30 citations

Pharmacy, Chemistry, Medicinal Chemistry +14