Katarzyna Kucwaj‐Brysz

SEL120-34A is a novel CDK8 inhibitor active in AML cells with high levels of serine phosphorylation of STAT1 and STAT5 transactivation domains

Tomasz Rzymski, Michał Mikuła, Eliza Żyłkiewicz et al. · Oncotarget · 2017 · 98 citations · Full text

Immunology, Lineage Commitment, Cancer Biology +17

In the search for a lead structure among series of potent and selective hydantoin 5‐<scp>HT</scp>₇R agents: The drug‐likeness in vitro study

Gniewomir Latacz, Annamaria Lubelska, Magdalena Jastrzębska‐Więsek et al. · Chemical Biology & Drug Design · 2017 · 47 citations · Full text

SAR-studies on the importance of aromatic ring topologies in search for selective 5-HT7 receptor ligands among phenylpiperazine hydantoin derivatives

Jadwiga Handzlik, Andrzej J. Bojarski, Grzegorz Satała et al. · European Journal of Medicinal Chemistry · 2014 · 41 citations · Full text

Aromatic Ring Topologies, Medicinal Chemistry, Drug Target +11

MF-8, a novel promising arylpiperazine-hydantoin based 5-HT7 receptor antagonist: In vitro drug-likeness studies and in vivo pharmacological evaluation

Gniewomir Latacz, Annamaria Lubelska, Magdalena Jastrzębska‐Więsek et al. · Bioorganic & Medicinal Chemistry Letters · 2018 · 39 citations · Full text

Synthesis and computer-aided SAR studies for derivatives of phenoxyalkyl-1,3,5-triazine as the new potent ligands for serotonin receptors 5-HT6

Wesam Ali, Małgorzata Więcek, Dorota Łażewska et al. · European Journal of Medicinal Chemistry · 2019 · 29 citations · Full text

Combinatorial Chemistry, Medicinal Chemistry, Derivative (Chemistry) +11