Heinz Stadtmüller

Start Selective and Rigidify: The Discovery Path toward a Next Generation of EGFR Tyrosine Kinase Inhibitors

Harald Engelhardt, Dietrich Böse, Mark Petronczki et al. · Journal of Medicinal Chemistry · 2019 · 145 citations · Full text

Medicine, Oncology, Pharmacology +17

A Novel RAF Kinase Inhibitor with DFG-Out–Binding Mode: High Efficacy in BRAF-Mutant Tumor Xenograft Models in the Absence of Normal Tissue Hyperproliferation

Irene C. Waizenegger, Anke Baum, Steffen Steurer et al. · Molecular Cancer Therapeutics · 2016 · 94 citations · Full text

Medicine, Oncology, Pharmacology +17

Stereoselective Preparation of Polyfunctional Cyclopentane Derivatives by Radical Nickel‐ or Palladium‐Catalyzed Carbozincations

Heinz Stadtmüller, Andrea Vaupel, Charles E. Tucker et al. · Chemistry - A European Journal · 1996 · 85 citations

Natural Sciences, Chemistry, Catalysis +10

Efficacy of the highly selective focal adhesion kinase inhibitor BI 853520 in adenocarcinoma xenograft models is linked to a mesenchymal tumor phenotype

Ulrich A. Hirt, Irene C. Waizenegger, Norbert Schweifer et al. · Oncogenesis · 2018 · 61 citations · Full text

Medicine, Oncology, Pharmacology +15

Stereoselective synthesis of polyfunctional di- and trisubstituted cyclopentane derivatives using a new palladium catalyzed cyclization.

Heinz Stadtmüller, Charles E. Tucker, Andrea Vaupel et al. · Tetrahedron Letters · 1993 · 52 citations

Natural Sciences, Chemistry, Catalysis +11