Vladimir A. Pavlyukovets

Structural insights into transient receptor potential vanilloid type 1 (TRPV1) from homology modeling, flexible docking, and mutational studies

Jin Hee Lee, Yoonji Lee, HyungChul Ryu et al. · Journal of Computer-Aided Molecular Design · 2011 · 71 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +17

Kinetics of Penetration Influence the Apparent Potency of Vanilloids on TRPV1

József Lázár, Derek C. Braun, Attila Tóth et al. · Molecular Pharmacology · 2006 · 32 citations

Medicine, Cell Biology, Pharmacology +10

Stereospecific High-affinity TRPV1 Antagonists: Chiral <i>N</i>-(2-Benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide Analogues

HyungChul Ryu, Mi-Kyoung Jin, Su Yeon Kim et al. · Journal of Medicinal Chemistry · 2007 · 30 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

α-Substituted N-(4-tert-butylbenzyl)-N′-[4-(methylsulfonylamino)benzyl]thiourea analogues as potent and stereospecific TRPV1 antagonists

Jae-Uk Chung, Su Yeon Kim, Ju‐Ok Lim et al. · Bioorganic & Medicinal Chemistry · 2007 · 26 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +4

Analysis of structure–activity relationships for the ‘A-region’ of N-(4-t-butylbenzyl)-N′-[4-(methylsulfonylamino)benzyl]thiourea analogues as TRPV1 antagonists

Jeewoo Lee, Sang-Uk Kang, Min-Jung Kil et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 24 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12