Concepedia
Statistics
Publications
7
Citations
274
H-Index
Active since
1990
Affiliations
Servier (France)(Current)
Inserm
Institut des Hautes Études Scientifiques
Patrick Hautefaye is an author at Servier (France) specializing in pharmacology, medicine, and drug discovery.
Top concepts
PharmacologyMedicineBiochemistryDrug DiscoveryEngineeringNatural SciencesOrganic ChemistryMedicinal ChemistryBiomolecular EngineeringOncology
Publications per year
1990–2011
New .alpha.-amino phosphonic acid derivatives of vinblastine: chemistry and antitumor activity
Gilbert Lavielle, Patrick Hautefaye, Corinne Schaeffer et al. · Journal of Medicinal Chemistry · 1991 · 127 citations
Medicinal Chemistry, Derivative (Chemistry), Bioorganic Chemistry +13
Synthesis and pharmacological evaluation of novel non-lactone analogues of camptothecin
Patrick Hautefaye, B. CIMETIERE, Alain St. Pierre et al. · Bioorganic & Medicinal Chemistry Letters · 2003 · 59 citations
Biochemistry, Medicine, Novel Non-lactone Analogues +5
Novel Stable Camptothecin Derivatives Replacing the E-Ring Lactone by a Ketone Function Are Potent Inhibitors of Topoisomerase I and Promising Antitumor Drugs
Amélie Lansiaux, Stéphane Léonce, Laurence Kraus‐Berthier et al. · Molecular Pharmacology · 2007 · 31 citations
Substituent control in the synthesis of azetidines and pyrrolidines by N-tosyl-oxiraneethylamines base-mediated cyclization.
J. Moulines, J.‐P. BATS, Patrick Hautefaye et al. · Tetrahedron Letters · 1993 · 21 citations
Engineering, Substituent Control, Diversity-oriented Synthesis +6
A convenient route to functionalized 3-amino-N-methylfuro[3,2-b]pyridine-2-carboxamides
Anne Bretéché, Pascal Marchand, Marie‐Renée Nourrisson et al. · Tetrahedron · 2011 · 14 citations
Engineering, Convenient Route, Organic Chemistry +2
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