Yannick Aussagues

Design, Synthesis and Biological Evaluation of 4‐Amino‐<i>N</i>‐(4‐aminophenyl)benzamide Analogues of Quinoline‐Based SGI‐1027 as Inhibitors of DNA Methylation

Elodie Rilova, Alexandre Erdmann, Christina Gros et al. · ChemMedChem · 2014 · 66 citations · Full text

Crystal Structure, Dna Methylation, Chemical Biology +20

Physalin B, a novel inhibitor of the ubiquitin-proteasome pathway, triggers NOXA-associated apoptosis

Isabelle Vandenberghe, Laurent Créancier, Stéphane Vispé et al. · Biochemical Pharmacology · 2008 · 62 citations

Triggers Noxa-associated Apoptosis, Physalin B, Protein Function +9

Rational Design of Bisubstrate-Type Analogues as Inhibitors of DNA Methyltransferases in Cancer Cells

Ludovic Halby, Yoann Menon, Elodie Rilova et al. · Journal of Medicinal Chemistry · 2017 · 56 citations · Full text

Anticancer activity of koningic acid and semisynthetic derivatives

Nicolas J. Rahier, Nicolas Molinier, Christophe Long et al. · Bioorganic & Medicinal Chemistry · 2015 · 37 citations

Medicinal Chemistry, Chemoprevention Strategy, Medicine +5

High-Throughput Bioluminescence Screening of Ubiquitin-Proteasome Pathway Inhibitors from Chemical and Natural Sources

Fréderic Ausseil, Arnaud Samson, Yannick Aussagues et al. · SLAS DISCOVERY · 2006 · 26 citations · Full text