Derick D. Winkle

Development of a Scalable Process for CI-1034, an Endothelin Antagonist

Thomas E. Jacks, Daniel T. Belmont, Christopher A. Briggs et al. · Organic Process Research & Development · 2004 · 55 citations

Organic Chemistry, Pharmacotherapy, Chemistry +18

Suzuki Reaction of a Diarylborinic Acid:  One-Pot Preparation and Cross-Coupling of Bis(3,5-dimethylphenyl)borinic Acid

Derick D. Winkle, Kevin M. Schaab · Organic Process Research & Development · 2001 · 31 citations

3,5-Dimethylphenylmagnesium Bromide Reacts, Chemical Engineering, Borinic Acid +11

Diastereoselective, large scale synthesis of β-amino acids via asymmetric enamide hydrogenation as α2δ ligands for the treatment of generalized anxiety disorder and insomnia

Javier Magano, Brian G. Conway, Daniel M. Bowles et al. · Tetrahedron Letters · 2009 · 22 citations

Enantioselective Synthesis, Large Scale Synthesis, Psychiatry +8

Tandem Transformations Involving Allylic Silanes. 2. Highly Diastereoselective Substitutions Involving [(Trialkylsilyl)methyl]cyclohexene Derivatives with Aldehydes. Synthetic Studies on the Problem of Lewis Acid-Promoted Protodesilylation and Enolization

Michael G. Organ, Derick D. Winkle, John C. Huffmann · The Journal of Organic Chemistry · 1997 · 20 citations

Diastereoselective, large-scale synthesis of β-amino acids via asymmetric aza-Michael addition as α2δ ligands for the treatment of generalized anxiety disorder and insomnia

Javier Magano, Daniel M. Bowles, Brian G. Conway et al. · Tetrahedron Letters · 2009 · 19 citations

Combinatorial Chemistry, Generalized Anxiety Disorder, Medicine +7