Synthesis and Immunosuppressive Activity of Novel Prodigiosin Derivatives

Roberto D’Alessio, Alberto Bargiotti, Orlando Carlini, +10

Journal of Medicinal Chemistry

Cdc7 Kinase Inhibitors: Pyrrolopyridinones as Potential Antitumor Agents. 1. Synthesis and Structure–Activity Relationships

Ermes Vanotti, Raffaella Amici, Alberto Bargiotti, +20

Journal of Medicinal Chemistry

Molecular BiologyStructure–activity RelationshipsPharmaceutical ChemistryMolecular PharmacologyMedicinal Chemistry +14

First Cdc7 Kinase Inhibitors: Pyrrolopyridinones as Potent and Orally Active Antitumor Agents. 2. Lead Discovery

Maria Menichincheri, Alberto Bargiotti, Jens Berthelsen, +28

Journal of Medicinal Chemistry

Molecular BiologyPharmacotherapyCell CycleTumor BiologyMolecular Pharmacology +15

Cdc7 Kinase Inhibitors: 5-Heteroaryl-3-Carboxamido-2-Aryl Pyrroles as Potential Antitumor Agents. 1. Lead Finding

Maria Menichincheri, Clara Albanese, Cristina Alli, +33

Journal of Medicinal Chemistry

Compound 18Lead IdentificationPharmaceutical ChemistryTumor BiologyMolecular Pharmacology +17

Catecholic Flavonoids Acting as Telomerase Inhibitors

Maria Menichincheri, Dario Ballinari, Alberto Bargiotti, +10

Journal of Medicinal Chemistry

Novel tumor-targeted RGD peptide–camptothecin conjugates: Synthesis and biological evaluation

Alma Dal Pozzo, Minghong Ni, Emiliano Esposito, +11

Bioorganic & Medicinal Chemistry

Drug DiscoveryBioconjugationPeptide TherapeuticPeptide SynthesisPeptide Therapeutics +3

A mild and stereospecific conversion of vicinal diols into olefins

Stephen Hanessian, Alberto Bargiotti, M. Larue

Tetrahedron Letters

EngineeringAlkene MetathesisOrganic ChemistryStereoselective SynthesisVicinal Diols +2

Cell Division Cycle 7 Kinase Inhibitors: 1<i>H</i>-Pyrrolo[2,3-<i>b</i>]pyridines, Synthesis and Structure−Activity Relationships

Antonella Ermoli, Alberto Bargiotti, Maria Gabriella Brasca, +16

Journal of Medicinal Chemistry

In vivo anti-tumour activity of FCE 23762, a methoxymorpholinyl derivative of doxorubicin active on doxorubicin-resistant tumour cells

Marina Ripamonti, Gabriella Pezzoni, Enrico Pesenti, +6

British Journal of Cancer

Tumor BiologyMedicinal ChemistryDrug TargetingDoxorubicin-resistant Tumour CellsVivo Anti-tumour Activity +9

Stereocontrolled glycosidation of daunomycinone. Synthesis and biological evaluation of 6-hydroxy-L-arabino analogues of antitumor anthracyclines

Federico Arcamone, Alberto Bargiotti, Giuseppe Cassinelli, +6

Journal of Medicinal Chemistry

Pharmaceutical ScienceBioorganic ChemistryGlycobiologyAltmetric Attention ScorePharmacotherapy +18