Laurent Dubois

Reactivity of 2,3-Aziridino-2,3-dideoxy-D-lyxono-.gamma.-lactone Derivatives, Rigid Analogs of Aziridine-2-carboxylic Esters, toward Soft and Hard Nucleophiles: Control of Lactone vs Aziridine Ring Opening and C-2 vs C-3 Regioselectivity

Philippe Dauban, Laurent Dubois, Marie Elise Tran Huu Dau et al. · The Journal of Organic Chemistry · 1995 · 65 citations

2,3-Aziridino-2,3-dideoxy-d-lyxono-.gamma.-lactone Derivatives, Engineering, Aziridine Ring Opening +10

Preparation of .beta.-substituted tryptophan derivatives: comparison of the reactivity of N-methylindole toward aziridine-2-lactones and aziridine-2-carboxylic esters and interpretation of results using MNDO calculations

Laurent Dubois, Anita Mehta, Emmanuelle Tourette et al. · The Journal of Organic Chemistry · 1994 · 60 citations

Medicinal Chemistry, Derivative (Chemistry), Derivatives +15

Stereocontrolled synthesis of aziridine-2-lactones from d-ribose and d-lyxose

Laurent Dubois, Robert H. Dodd · Tetrahedron · 1993 · 39 citations

Engineering, Organic Chemistry, Stereoselective Synthesis +4

Synthetic Routes to 4-Amino-3-carboxy-.beta.-carboline Derivatives: Incidental Formation of Novel Furo[3,4-c]-.beta.-carbolin-2-ones Displaying High Affinities for the Benzodiazepine Receptor

Gilbert Dorey, Laurent Dubois, Lia Prdo Prado de Carvalho et al. · Journal of Medicinal Chemistry · 1995 · 19 citations

Preparation of the (R) and (S) enantiomers of 10-hydroxymethylfuro[3,4-c]-β-carboline-2(10H)one, the first example of a benzodiazepine receptor ligand of the β-carboline family having a stereogenic center

Laurent Dubois, Gilbert Dorey, Pierre Potìer et al. · Tetrahedron Asymmetry · 1995 · 17 citations

Molecular Pharmacology, Benzodiazepine Receptor Ligand, Medicine +8