Gregory A. Gfesser

4-(2-[2-(2(<i>R</i>)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and Related 2-Aminoethylbenzofuran H₃ Receptor Antagonists Potently Enhance Cognition and Attention

Marlon Cowart, Ramin Faghih, Michael P. Curtis et al. · Journal of Medicinal Chemistry · 2004 · 121 citations · Full text

Receptor Antagonists, Psychopharmacology, Pharmacotherapy +17

Synthesis and SAR of 5-Amino- and 5-(Aminomethyl)benzofuran Histamine H₃Receptor Antagonists with Improved Potency

Minghua Sun, Chen Zhao, Gregory A. Gfesser et al. · Journal of Medicinal Chemistry · 2005 · 62 citations · Full text

Discovery of 4-(5-(4-Chlorophenyl)-2-methyl-3-propionyl-1<i>H</i>-pyrrol-1-yl)benzenesulfonamide (A-867744) as a Novel Positive Allosteric Modulator of the α7 Nicotinic Acetylcholine Receptor

Ramin Faghih, Sujatha M. Gopalakrishnan, Jens Halvard Grønlien et al. · Journal of Medicinal Chemistry · 2009 · 53 citations · Full text

5-(3-Bromophenyl)-7-(6-morpholin-4-ylpyridin-3-yl)pyrido[2,3-d]pyrimidin-4-ylamine: structure–activity relationships of 7-substituted heteroaryl analogs as non-nucleoside adenosine kinase inhibitors

Mark A. Matulenko, Chih‐Hung Lee, Meiqun Jiang et al. · Bioorganic & Medicinal Chemistry · 2005 · 48 citations

Molecular Pharmacology, Medicinal Chemistry, Biochemistry +13

Structure–activity relationships of arylbenzofuran H3 receptor antagonists

Gregory A. Gfesser, Ramin Faghih, Youssef L. Bennani et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 47 citations

Molecular Pharmacology, Biochemistry, Medicine +5