Christian Dubiella

Statistics

Publications

Citations

457

H-Index

Active since

2014

Affiliations

Center for Integrated Protein Science Munich(Current)

Technical University of Munich

Saarland University

Weizmann Institute of Science

Christian Dubiella is an author at Center for Integrated Protein Science Munich specializing in enzyme inhibition, drug discovery, and medicinal chemistry.

ORCID

Publications per year

2014–2022

Publications

Sulfopin is a covalent inhibitor of Pin1 that blocks Myc-driven tumors in vivo

Christian Dubiella, Benika J. Pinch, Kazuhiro Koikawa et al. · Nature Chemical Biology · 2021 · 148 citations · Full text

Medicine, Molecular Biology, Oncology +14

Selective Inhibition of the Immunoproteasome by Ligand‐Induced Crosslinking of the Active Site

Christian Dubiella, Haissi Cui, Malte Gersch et al. · Angewandte Chemie International Edition · 2014 · 91 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12

Systematic Comparison of Peptidic Proteasome Inhibitors Highlights the α‐Ketoamide Electrophile as an Auspicious Reversible Lead Motif

Martin Stein, Haissi Cui, Philipp Beck et al. · Angewandte Chemie International Edition · 2014 · 83 citations

Life Sciences, Biochemistry, Medicinal Chemistry +15

Macyranones: Structure, Biosynthesis, and Binding Mode of an Unprecedented Epoxyketone that Targets the 20S Proteasome

Lena Keller, Alberto Plaza, Christian Dubiella et al. · Journal of the American Chemical Society · 2015 · 40 citations

Life Sciences, Biochemistry, Molecular Biology +13

Selective Inhibition of the Immunoproteasome by Structure‐Based Targeting of a Non‐catalytic Cysteine

Christian Dubiella, Regina Baur, Haissi Cui et al. · Angewandte Chemie International Edition · 2015 · 29 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

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