Frank Marsilio

(2<i>R</i>)-4-Oxo-4-[3-(Trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-<i>a</i>]pyrazin- 7(8<i>H</i>)-yl]-1-(2,4,5-trifluorophenyl)butan-2-amine:  A Potent, Orally Active Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type 2 Diabetes

Dooseop Kim, Liping Wang, Maria Beconi et al. · Journal of Medicinal Chemistry · 2004 · 808 citations · Full text

Catalytic properties and inhibition of proline-specific dipeptidyl peptidases II, IV and VII

Barbara Leiting, KellyAnn D. Pryor, Joseph K. Wu et al. · Biochemical Journal · 2003 · 181 citations · Full text

Proteomic Technology, Molecular Pharmacology, Catalytic Constants +15

Substituted piperazines as novel dipeptidyl peptidase IV inhibitors

Linda Brockunier, Jiafang He, Lawrence F. Colwell et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 97 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Medicine +6

Discovery of potent and selective β-homophenylalanine based dipeptidyl peptidase IV inhibitors

Jinyou Xu, Hyun Ok, Edward J. Gonzalez et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 76 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Biochemistry +7

Discovery of potent and selective phenylalanine based dipeptidyl peptidase IV inhibitors

Jinyou Xu, Lan Wei, Robert J. Mathvink et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 68 citations

Medicinal Chemistry, Biochemistry, Natural Sciences +9